发明名称 |
FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS |
摘要 |
Compounds having the formula (I), and enantiomers, and diastereomers, pharmaceutically-acceptable salts, and hydrates, thereof, (I) are useful as kinase modulators, including MK2 modulation, wherein one of E and F is a nitrogen atom and the other of E and F is a carbon atom, and Z is N or CR3, and R1, R2, R3, X and Y are as defined herein. |
申请公布号 |
CA2623369(C) |
申请公布日期 |
2014.11.18 |
申请号 |
CA20062623369 |
申请日期 |
2006.09.22 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
VACCARO, WAYNE;CHEN, ZHONG;DODD, DHARMPAL S.;HUYNH, TRAM N.;LIN, JAMES;LIU, CHUNJIAN;MUSSARI, CHRISTOPHER P.;TOKARSKI, JOHN S.;TORTOLANI, DAVID R.;WROBLESKI, STEPHEN T. |
分类号 |
C07D487/04;A61K31/437;A61P29/00 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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