发明名称 COMPOSTOS, PROCESSO DE FABRICAÇÃO DESTES, COMPOSIÇÃO FARMACÊUTICA QUE OS CONTÉM, MÉTODO DE TRATAMENTO E/OU PREVENÇÃO DE DOENÇAS QUE SÃO ASSOCIADAS A MODULAÇÃO DE RECEPTORES DE SST SUBTIPO 5 E USO DOS COMPOSTOS.
摘要 This invention relates to compounds of the formula wherein A, R1 to R3 are as defined in the claims and G is benzoimidazole, quinoxaline, benzotriazole, dihydro-imidazo[4,5-c]pyridinone and dihydro-isoindolone group as defined in the specification, and pharmaceutically acceptable salts thereof. The invention further relates to pharmaceutical compositions containing such compounds, to a process for their preparation and to their use for the treatment and/or prevention of diseases which are associated with the modulation of SST receptors subtype 5 such as diabetes mellitus.
申请公布号 BRPI0809981(A2) 申请公布日期 2014.10.14
申请号 BR2008PI09981 申请日期 2008.03.26
申请人 F. HOFFMANN-LA ROCHE AG 发明人 KONRAD BLEICHER;PETER MOHR;RAINER E. MARTIN;ANDREAS D. CHRIST
分类号 C07D401/04;A61K31/454;A61P5/50;C07D401/14;C07D405/14;C07D471/04 主分类号 C07D401/04
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