发明名称 Heterocyclic substituted pyridine derivatives and antifungal agent containing same
摘要 <p>An object of the present invention is to provide an antifungal agent which has excellent antifungal effects and is superior in terms of its physical properties, safety and metabolic stability. According to the present invention, there is disclosed a compound or a pharmaceutically acceptable salt thereof, the compound being selected from the group consisting of 3-(3-(4-(pyridin-2-yloxymethyl)-benzyl)-isoxazol-5-yl)-pyridin-2-ylamine; 3-(3-(4-(Pyridin-2-ylmethoxy)-benzyl)-isoxazol-5-yl)-pyridin-2-ylamine; 3-(3-(4-pyridin-2-yloxymethyl)-benzyl)-isoxazol-5-yl)-pyridine-2,6-diamine; 3-(3-(6-benzyloxy-pyridin-3-ylmethyl)-isoxazol-5-yl)-pyridin-2,6-diamine; and 3-(1-(4-(pyridin-2-yloxymethyl)-benzyl)-1H-pyrazol-4-yl)-pyridin-2-ylamine.</p>
申请公布号 EP2628738(B1) 申请公布日期 2014.09.03
申请号 EP20120193373 申请日期 2006.10.30
申请人 EISAI R&D MANAGEMENT CO., LTD. 发明人 TANAKA, KEIGO;INOUE, SATOSHI;MURAI, NORIO;MATSUKURA, MASAYUKI;NAKAMOTO, KAZUTAKA;SHIROTORI, SHUJI;ABE, SHINYA
分类号 C07D401/04;A61K31/4439;A61K31/444;A61P31/10;C07D401/14;C07D413/04;C07D413/14 主分类号 C07D401/04
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