发明名称 |
QUINAZOLINE DERIVATIVES AS PI3K MODULATORS |
摘要 |
<p>The invention relates to substituted quinazoline derivative of the formula (I), wherein A, X1, X2, X3, X4 and R5 are as defined in the description. Such compounds are suitable for the treatment of a disorder or disease which is mediated by the activity of the PI3K enzymes.</p> |
申请公布号 |
EP2768813(A1) |
申请公布日期 |
2014.08.27 |
申请号 |
EP20120791859 |
申请日期 |
2012.10.19 |
申请人 |
NOVARTIS AG |
发明人 |
FURET, PASCAL;HEBACH, CHRISTINA;HÖGENAUER, KLEMENS;HOLLINGWORTH, GREGORY;LEWIS, IAN;SMITH, ALEXANDER, BAXTER;SOLDERMANN, NICOLAS;STAUFFER, FRÉDÉRIC;WOLF, ROMAIN;ZECRI, FRÉDÉRIC |
分类号 |
C07D239/74;A61K31/517;A61P11/00;A61P29/00;A61P35/00;A61P37/00;C07D401/04;C07D401/14;C07D403/04;C07D403/14;C07D413/14;C07D487/08 |
主分类号 |
C07D239/74 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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