发明名称 |
4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1 H-imidazo(4,5-c)quinolin-7-yl)-3,5-dimethylisoxazole and its use as bromodomain inhibitor |
摘要 |
Novel quinoline compounds of formula (I), pharmaceutical compositions containing such compounds and their use in therapy, as bromodomain inhibitors. |
申请公布号 |
AU2012296914(A1) |
申请公布日期 |
2014.02.13 |
申请号 |
AU20120296914 |
申请日期 |
2012.08.15 |
申请人 |
GLAXOSMITHKLINE LLC |
发明人 |
DEMONT, EMMANUEL HUBERT;JONES, KATHERINE LOUISE;WATSON, ROBERT J. |
分类号 |
C07D471/04;A61K31/4745;A61P29/00;A61P37/00 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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