发明名称 PROCESSES FOR PREPARING TUBULYSINS
摘要 Tubulysins are a series of naturally occurring cytotoxic agents that are of interest as anticancer therapeutic agents. Processes and intermediates useful for preparing naturally occurring and non-naturally occurring tubulysins and analogs and derivatives thereof are described.
申请公布号 EP2600866(A4) 申请公布日期 2013.12.11
申请号 EP20110815381 申请日期 2011.08.05
申请人 ENDOCYTE, INC. 发明人 VLAHOV, IONTCHO, RADOSLAVOV;GROANING, MICHAEL;KLEINDL, PAUL, JOSEPH;SANTHAPURAM, HARI KRISHNA, R.;YOU, FEI;WANG, YU;XU, LE-CUN;STANFORD, KATHERYN, MARIE;RITTER, ALLEN;LEAMON, CHRISTOPHER, PAUL
分类号 C07D417/12;A61K31/445;A61K31/4535;A61P35/00 主分类号 C07D417/12
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