Tubulysins are a series of naturally occurring cytotoxic agents that are of interest as anticancer therapeutic agents. Processes and intermediates useful for preparing naturally occurring and non-naturally occurring tubulysins and analogs and derivatives thereof are described.
申请公布号
EP2600866(A4)
申请公布日期
2013.12.11
申请号
EP20110815381
申请日期
2011.08.05
申请人
ENDOCYTE, INC.
发明人
VLAHOV, IONTCHO, RADOSLAVOV;GROANING, MICHAEL;KLEINDL, PAUL, JOSEPH;SANTHAPURAM, HARI KRISHNA, R.;YOU, FEI;WANG, YU;XU, LE-CUN;STANFORD, KATHERYN, MARIE;RITTER, ALLEN;LEAMON, CHRISTOPHER, PAUL