发明名称 |
NOVEL beta-LACTAMASE INHIBITOR AND METHOD FOR PRODUCING SAME |
摘要 |
Currently available beta-lactamase inhibitors have an inadequate effect against beta-lactamases, which continue to increase constantly. There is a need for novel beta-lactamase inhibitors which can be used in the treatment of bacterial infections caused by resistant bacteria that are currently difficult to treat and that produce: class C beta-lactamase; extended-spectrum beta-lactamase (ESBL) belonging to classes A and D; KPC-2, which decomposes even carbapenem, the last bastion of beta-lactam antibiotics, belonging to class A; and the like. Provided are a compound shown by formula (I), a method for producing the same, a beta-lactamase inhibitor, and a method for treating bacterial infections. |
申请公布号 |
WO2013180197(A1) |
申请公布日期 |
2013.12.05 |
申请号 |
WO2013JP64971 |
申请日期 |
2013.05.30 |
申请人 |
MEIJI SEIKA PHARMA CO., LTD. |
发明人 |
ABE, TAKAO;FURUUCHI, TAKESHI;SAKAMAKI, YOSHIAKI;INAMURA, SEIICHI;MORINAKA, AKIHIRO |
分类号 |
C07D471/08;A61K31/439;A61K31/444;A61K31/4545;A61K31/5377;A61P31/04;A61P43/00;C07D211/60 |
主分类号 |
C07D471/08 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|