发明名称 BENZODIAZEPINE DERIVATIVE FOR THE TREATMENT OF HEMATOPOIETIC NEOPLASM AND LEUKEMIA
摘要 A method and medicament for treating mixed lineage leukemia; translocated mixed lineage leukemia; translocated mixed lineage leukemia based acute myelogenous leukemia; translocated mixed lineage leukemia based acute lymphoid leukemia; a non-MLL based chronic myeloproloferative disorder, or non-MLL based acoute lymphoid leukemia is provided, wherein the active agent used is the GSK-3 inhibitor 7-(2,5-dihydro-4-imidazo[1,2-a]pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4-tetrahydro-2-(1-piperidinylcarbonyl)pyrrolo[3,2,1-jk]-[1,4]benzodiazepine or a pharmaceutically acceptable salt or salvate thereof.
申请公布号 EA018933(B1) 申请公布日期 2013.11.29
申请号 EA20110071243 申请日期 2010.04.08
申请人 ELI LILLY AND COMPANY 发明人 CHEDID MARCIO
分类号 A61K31/5517;A61P35/02 主分类号 A61K31/5517
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