发明名称 TETRAHYDROPYRROLOTHIAZINE COMPOUNDS
摘要 The present invention provides compounds of Formula I: wherein A is selected from the group consisting of; (a), (b), (c) and (d), R1 is H or F; R2 is H, -CH2OH, C1-C3 alkyl, (e), or (f);; R3 is H, F, or CN; R4 is H, F; or CN; and R5 is H, -CH3, or -OCH3; or a pharmaceutically acceptable salt thereof.
申请公布号 WO2013151832(A1) 申请公布日期 2013.10.10
申请号 WO2013US33959 申请日期 2013.03.27
申请人 ELI LILLY AND COMPANY 发明人 BECK, JAMES PETER;GREEN, STEVEN JAMES;LOPEZ, JOSE EDUARDO;MATHES, BRIAN MICHAEL;MERGOTT, DUSTIN JAMES;PORTER, WARREN JAYE;RANKOVIC, ZORAN;SHI, YUAN;WATSON, BRIAN MORGAN;WINNEROSKI, JR., LEONARD LARRY
分类号 C07D513/04;A61K31/407;A61P25/28 主分类号 C07D513/04
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