发明名称 |
TETRAHYDROPYRROLOTHIAZINE COMPOUNDS |
摘要 |
The present invention provides compounds of Formula I: wherein A is selected from the group consisting of; (a), (b), (c) and (d), R1 is H or F; R2 is H, -CH2OH, C1-C3 alkyl, (e), or (f);; R3 is H, F, or CN; R4 is H, F; or CN; and R5 is H, -CH3, or -OCH3; or a pharmaceutically acceptable salt thereof. |
申请公布号 |
WO2013151832(A1) |
申请公布日期 |
2013.10.10 |
申请号 |
WO2013US33959 |
申请日期 |
2013.03.27 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
BECK, JAMES PETER;GREEN, STEVEN JAMES;LOPEZ, JOSE EDUARDO;MATHES, BRIAN MICHAEL;MERGOTT, DUSTIN JAMES;PORTER, WARREN JAYE;RANKOVIC, ZORAN;SHI, YUAN;WATSON, BRIAN MORGAN;WINNEROSKI, JR., LEONARD LARRY |
分类号 |
C07D513/04;A61K31/407;A61P25/28 |
主分类号 |
C07D513/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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