发明名称 Preparation of (R)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide and (S)-N-3,4-difluoro-2(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide
摘要 The present invention relates to the preparation of (R)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide and (S)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide.
申请公布号 US8513443(B2) 申请公布日期 2013.08.20
申请号 US201013386519 申请日期 2010.07.10
申请人 MADERNA ANDREAS;VERNIER JEAN-MICHEL;ARDEA BIOSCIENCES, INC. 发明人 MADERNA ANDREAS;VERNIER JEAN-MICHEL
分类号 C07D317/10 主分类号 C07D317/10
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