发明名称 |
Preparation of (R)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide and (S)-N-3,4-difluoro-2(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide |
摘要 |
The present invention relates to the preparation of (R)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide and (S)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide.
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申请公布号 |
US8513443(B2) |
申请公布日期 |
2013.08.20 |
申请号 |
US201013386519 |
申请日期 |
2010.07.10 |
申请人 |
MADERNA ANDREAS;VERNIER JEAN-MICHEL;ARDEA BIOSCIENCES, INC. |
发明人 |
MADERNA ANDREAS;VERNIER JEAN-MICHEL |
分类号 |
C07D317/10 |
主分类号 |
C07D317/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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