发明名称 CARBOXAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS
摘要 The present invention provides compounds that are inhibitors of voltage-gated sodium channels (Nav), in particular Nav 1.7, and are therefore useful for the treatment of diseases treatable by inhibition of these channels, in particular, chronic pain disorders. Also provided are pharmaceutical compositions containing such compounds and processes for preparing such compounds.
申请公布号 US2013131035(A1) 申请公布日期 2013.05.23
申请号 US201113575912 申请日期 2011.02.16
申请人 BREGMAN HOWARD;BUCHANAN JOHN L.;CHAKKA NAGASREE;DIMAURO ERIN F.;DU BINGFAN;NGUYEN HANH NHO;ZHENG XIAO MEI;AMGEN INC. 发明人 BREGMAN HOWARD;BUCHANAN JOHN L.;CHAKKA NAGASREE;DIMAURO ERIN F.;DU BINGFAN;NGUYEN HANH NHO;ZHENG XIAO MEI
分类号 C07D471/10;C07D251/48;C07D401/04;C07D403/04 主分类号 C07D471/10
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