发明名称 |
Pyrazole [3, 4-B] pyridine Raf inhibitors |
摘要 |
Compounds of Formula I are useful for inhibition of Raf kinases. Methods of using compounds of Formula I and stereoisomers, tautomers, prodrugs and pharmaceutically acceptable salts thereof, for in vitro, in situ, and in vivo diagnosis, prevention or treatment of such disorders in mammalian cells, or associated pathological conditions are disclosed. |
申请公布号 |
US8394795(B2) |
申请公布日期 |
2013.03.12 |
申请号 |
US20090920050 |
申请日期 |
2009.02.27 |
申请人 |
AHRENDT KATERI A.;BUCKMELTER ALEXANDRE J.;DE MEESE JASON;GRINA JONAS;HANSEN JOSHUA D.;LAIRD ELLEN R.;LUNGHOFER PAUL;MORENO DAVID;NEWHOUSE BRAD;REN LI;SEO JEONGBEOB;TIAN HONGQI;WENGLOWSKY STEVEN MARK;FENG BAINIAN;GUNZNER JANET;MALESKY KIM;MATHIEU SIMON;RUDOLPH JOACHIM;WEN ZHAOYANG;YOUNG WENDY B.;ARRAY BIOPHARMA INC.;GENENTECH, INC. |
发明人 |
AHRENDT KATERI A.;BUCKMELTER ALEXANDRE J.;DE MEESE JASON;GRINA JONAS;HANSEN JOSHUA D.;LAIRD ELLEN R.;LUNGHOFER PAUL;MORENO DAVID;NEWHOUSE BRAD;REN LI;SEO JEONGBEOB;TIAN HONGQI;WENGLOWSKY STEVEN MARK;FENG BAINIAN;GUNZNER JANET;MALESKY KIM;MATHIEU SIMON;RUDOLPH JOACHIM;WEN ZHAOYANG;YOUNG WENDY B. |
分类号 |
A61K31/535;A61K31/44;C07D413/14;C07D471/04 |
主分类号 |
A61K31/535 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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