发明名称 Process for the preparation of dihydroquinazolines
摘要 The present invention relates to a process for the preparation of dihydroquinazolines, for example, methyl (S)-{8-fluoro-2-[4-(3-methoxyphenyl)piperazin-1-yl]-3-[2-methoxy-5-(trifluoro -methyl)-phenyl]-3,4-dihydroquinazolin-4-yl}acetate (2S,3S)-2,3-bis[(4-methylbenzoyl) -oxy]succinic acid salt, which are used for the production of antiviral medicaments.
申请公布号 US8372972(B2) 申请公布日期 2013.02.12
申请号 US201113308418 申请日期 2011.11.30
申请人 AICURIS GMBH & CO. KG;GOOBETAEN KAETHE;KUHN OLIVER;BERWE MATHIAS;KRUGER JOACHIM;MILITZER HANS-CHRISTIAN 发明人 GOOBETAEN KAETHE;KUHN OLIVER;BERWE MATHIAS;KRUGER JOACHIM;MILITZER HANS-CHRISTIAN
分类号 C07D239/72 主分类号 C07D239/72
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