发明名称 HIV INTEGRASE INHIBITORY OXOISOINDOLINE SULFONAMIDES
摘要 Novel oxoisoindoline sulfonamide integrase inhibitors are useful to inhibit HIV activity, and are therefore suitable for treatment or prophylaxis of HIV infection, for example in the treatment or prevention of AIDS. In particular embodiments, the inhibitors are oxoisoindoline-4- sulfonamides, such as 6,7- dihydroxy- 1 -oxoisomdolirie-4-sulfonamides.
申请公布号 WO2013016441(A1) 申请公布日期 2013.01.31
申请号 WO2012US48169 申请日期 2012.07.25
申请人 THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES;ZHAO, XUE, ZHI;HUGHES, STEPHEN, H.;VU, BAO-HAN, CHRISTIE;SMITH, STEVEN;JOHNSON, BARRY;POMMIER, YVES;BURKE, TERRENCE, R., JR. 发明人 ZHAO, XUE, ZHI;HUGHES, STEPHEN, H.;VU, BAO-HAN, CHRISTIE;SMITH, STEVEN;JOHNSON, BARRY;POMMIER, YVES;BURKE, TERRENCE, R., JR.
分类号 C07D209/46;A61K31/4035;A61P31/18;C07D401/12;C07D403/14;C07D515/04 主分类号 C07D209/46
代理机构 代理人
主权项
地址