发明名称 METHOD FOR THE PRODUCTION OF AMINO CROTONYL COMPOUNDS
摘要 The invention relates to a process for preparing a compound of general formula (VII): (see formula VII) comprising the following synthesis steps: a) reacting a compound of general formula (V) (see formula V) in suitable solvents after corresponding activation with di-(C1-4-alkyl)-phosphonoacetic acid; and b) reacting the resulting compound of general formula (VI) (see formula VI) with an aldehyde of formula (see formula a) or a corresponding aldehyde equivalent using suitable organic or inorganic bases.
申请公布号 CA2541928(C) 申请公布日期 2012.12.11
申请号 CA20042541928 申请日期 2004.10.12
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH 发明人 RALL, WERNER;SOYKA, RAINER;KULINNA, CHRISTIAN;SCHNAUBELT, JUERGEN;SIEGER, PETER
分类号 C07D405/12;A61K31/505;A61K31/517 主分类号 C07D405/12
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