发明名称 PIPERIDINE DERIVATIVES AND COMPOSITIONS FOR THE INHIBITION OF NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE (NAMPT)
摘要 The present invention relates to compounds and compositions for the inhibition of NAMPT, their synthesis, applications and antidotes. An illustrative compound of the invention is shown below: Formula (I)
申请公布号 CA2834745(A1) 申请公布日期 2012.11.15
申请号 CA20112834745 申请日期 2011.09.02
申请人 FORMA TM, LLC 发明人 BAIR, KENNETH W.;BAUMEISTER, TIMM;BUCKMELTER, ALEXANDRE J.;CLODFELTER, KARL H.;HAN, BINGSONG;KUNTZ, JUDITH D.;LIN, JIAN;REYNOLDS, DOMINIC J.;SMITH, CHASE C.;WANG, ZHONGGUO;ZHENG, XIAOZHANG
分类号 C07D215/48;A61K31/4523;A61P11/00;A61P11/06;A61P31/12;A61P31/18;A61P35/00;C07D471/04;C07D513/04;C07D519/00 主分类号 C07D215/48
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