发明名称 |
PYRROLO[2,3-d]PYRIMIDINE TROPOMYSIN-RELATED KINASE INHIBITORS |
摘要 |
The present invention relates to compounds of Formula (I) and their pharmaceutically acceptable salts, wherein the substituents are as described herein, and their use in medicine, in particular as Trk antagonists.
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申请公布号 |
US2012258950(A1) |
申请公布日期 |
2012.10.11 |
申请号 |
US201213439131 |
申请日期 |
2012.04.04 |
申请人 |
ANDREWS MARK DAVID;BAGAL SHARANJEET KAUR;GIBSON KARL RICHARD;OMOTO KIYOYUKI;RYCKMANS THOMAS;SKERRATT SARAH ELIZABETH;STUPPLE PAUL ANTHONY;PFIZER LIMITED |
发明人 |
ANDREWS MARK DAVID;BAGAL SHARANJEET KAUR;GIBSON KARL RICHARD;OMOTO KIYOYUKI;RYCKMANS THOMAS;SKERRATT SARAH ELIZABETH;STUPPLE PAUL ANTHONY |
分类号 |
A61K31/519;A61K31/52;A61P25/00;C07D473/00;C07D487/04 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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