发明名称 |
PROCESS FOR PREPARING DOCETAXEL AND ITS HYDRATE |
摘要 |
<p>Disclosed is a process of preparation of (2R,3S)-N-carboxy-3-phenylisoserine, N-tert-butyl ester, 13-ester with 5(P)-20-epoxy-l,2(a), 4,7(P), 10(ß), 13(a)-hexa hydroxyl tax-l l-en-9-one 4-acetate 2-benzoate (docetaxel) and its trihydrate (I).</p> |
申请公布号 |
WO2012131698(A1) |
申请公布日期 |
2012.10.04 |
申请号 |
WO2011IN00588 |
申请日期 |
2011.08.29 |
申请人 |
SHILPA MEDICARE LIMITED;SHRAWAT, VIMAL KUMAR;., VEERESHAPPA;PUROHIT, PRASHANT;RAFIUDDIN, . |
发明人 |
SHRAWAT, VIMAL KUMAR;., VEERESHAPPA;PUROHIT, PRASHANT;RAFIUDDIN, . |
分类号 |
C07D305/14;A61K31/337;A61P35/00 |
主分类号 |
C07D305/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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