| 发明名称 |
THIOPHENE OR THIAZOLE DERIVATIVES AND USE THEREOF AS PI3K INHIBITORS |
| 摘要 |
A compound of formula (I), wherein the values R1, R2, CY, Y1, Y2, X1, X2, and X3 are provided in the description, pharmaceutical compositions on a basis thereof, and their application for PI3K activity inhibition in patients, and proliferative, inflammatory or cardiovascular disorders treatment.
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| 申请公布号 |
GEP20125650(B) |
申请公布日期 |
2012.09.25 |
| 申请号 |
GE2009AP12065 |
申请日期 |
2009.06.17 |
| 申请人 |
MILLENNIUM PHARMACEUTICALS, INC. |
发明人 |
CARDIN, DAVID, P.;GAULIN, JEFFREY, L.;GREENSPAN, PAUL, D.;VYSKOCIL, STEPAN;XU, TIANLIN;RENOU, CHRISTELLE, C. |
| 分类号 |
C07D409/04;A61K31/4196;A61K31/427;A61K31/5377;C07D409/14;C07D417/04 |
主分类号 |
C07D409/04 |
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