发明名称 |
SELECTIVE LIGANDS FOR THE DOPAMINE 3 (D3) RECEPTOR AND METHODS OF USING THE SAME |
摘要 |
Potent and selective ligands for the dopamine 3 (D3) receptor are disclosed. The D3 receptor ligands have a structural formula: wherein R1 is C1-6 alkyl or C3-6cycloalkyl; or wherein R2 is substituted with one or two halogen(s) or OC1-3alkyl. |
申请公布号 |
US2012232118(A1) |
申请公布日期 |
2012.09.13 |
申请号 |
US201213406803 |
申请日期 |
2012.02.28 |
申请人 |
WANG SHAOMENG;CHEN JIANYONG;COLLINS GREGORY;LEVANT BETH;WOODS JAMES H.;UNIVERSITY OF KANSAS;THE REGENTS OF THE UNIVERSITY OF MICHIGAN |
发明人 |
WANG SHAOMENG;CHEN JIANYONG;COLLINS GREGORY;LEVANT BETH;WOODS JAMES H. |
分类号 |
A61K31/4245;A61K31/428;A61K31/4439;A61P3/00;A61P25/00;A61P25/08;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/30;A61P25/32;C07D277/82;C07D417/12 |
主分类号 |
A61K31/4245 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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