发明名称 |
PROCESS FOR PREPARING 5-FLUORO-1H-PYRAZOLO [3,4-B] PYRIDIN-3-AMINE AND DERIVATIVES THEREOF |
摘要 |
The present invention relates to a process for the synthesis of 5-fluoro-1H-pyrazolo[3,4-b]pyridin-3-amine in high yield and purity. The present invention also relates to processes for the synthesis of 5-fluoro-1H-pyrazolo[3,4-b]pyridin-3-amine derivatives. These processes are useful for preparing biologically active compounds, particularly certain GSK-3 inhibitors, or derivatives thereof.
|
申请公布号 |
US2012232275(A1) |
申请公布日期 |
2012.09.13 |
申请号 |
US201213347926 |
申请日期 |
2012.01.11 |
申请人 |
JIMENEZ JUAN-MIGUEL;COLLIER PHILIP;GREEN JEREMY;MILLER ANDREW;GAO HUAI;HAMON SYLVAIN LOIC JEAN-LUC;DROS ALBERT CORNELIS;VERTEX PHARMACEUTICALS INCORPORATED |
发明人 |
JIMENEZ JUAN-MIGUEL;COLLIER PHILIP;GREEN JEREMY;MILLER ANDREW;GAO HUAI;HAMON SYLVAIN LOIC JEAN-LUC;DROS ALBERT CORNELIS |
分类号 |
C07D471/04 |
主分类号 |
C07D471/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|