发明名称 3-AMINO-PYRIDINES AS GPBAR1 AGONISTS
摘要 <p>This invention relates to novel 3-aminopyridines of the formula (I) wherein B1, B2 and R1 to R6 are as defined in the description and in the claims, as well as pharmaceutically acceptable salts thereof. These compounds are GPBAR1 agonists and can be used as medicaments for the treatment of diseases such as type II diabetes.</p>
申请公布号 WO2012117000(A1) 申请公布日期 2012.09.07
申请号 WO2012EP53386 申请日期 2012.02.29
申请人 F. HOFFMANN-LA ROCHE AG;BISSANTZ, CATERINA;DEHMLOW, HENRIETTA;ERICKSON, SHAWN DAVID;KARNACHI, PRABHA SABA;KIM, KYUNGJIN;MARTIN, RAINERM, E.;MATTEI, PATRIZIO;OBST SANDER, ULRIKE;PIETRANICO-COLE, SHERRIE LYNN;RICHTER, HANS;ULLMER, CHRISTOPH 发明人 BISSANTZ, CATERINA;DEHMLOW, HENRIETTA;ERICKSON, SHAWN DAVID;KARNACHI, PRABHA SABA;KIM, KYUNGJIN;MARTIN, RAINERM, E.;MATTEI, PATRIZIO;OBST SANDER, ULRIKE;PIETRANICO-COLE, SHERRIE LYNN;RICHTER, HANS;ULLMER, CHRISTOPH
分类号 C07D213/75;A61K31/4418;A61K31/4433;C07D213/81;C07D213/82;C07D401/04;C07D401/12;C07D401/14;C07D405/04;C07D405/12;C07D413/04;C07D413/12;C07D417/04;C07D417/12;C07D491/107 主分类号 C07D213/75
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