发明名称 SUBSTITUTED [(5H-PYRROLO[2,1-c][1,4]BENZODIAZEPIN-11-YL)PIPERAZIN-1-YL]-2,2-DIMETHYLPROPANOIC ACID COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS
摘要 A dual H1/5-HT2A receptor antagonist of the formula: its uses, and methods for its preparation are described.
申请公布号 US2012202797(A1) 申请公布日期 2012.08.09
申请号 US201213357627 申请日期 2012.01.25
申请人 CAMP ANNE MARIE;GALLAGHER PETER THADDEUS;LEDGARD ANDREW JAMES;SANDERSON ADAM JAN;COATES DAVID ANDREW;ELI LILLY AND COMPANY 发明人 CAMP ANNE MARIE;GALLAGHER PETER THADDEUS;LEDGARD ANDREW JAMES;SANDERSON ADAM JAN;COATES DAVID ANDREW
分类号 A61K31/5517;A61P25/20;C07D487/04 主分类号 A61K31/5517
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