发明名称 |
SUBSTITUTED [(5H-PYRROLO[2,1-c][1,4]BENZODIAZEPIN-11-YL)PIPERAZIN-1-YL]-2,2-DIMETHYLPROPANOIC ACID COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS |
摘要 |
A dual H1/5-HT2A receptor antagonist of the formula: its uses, and methods for its preparation are described. |
申请公布号 |
US2012202797(A1) |
申请公布日期 |
2012.08.09 |
申请号 |
US201213357627 |
申请日期 |
2012.01.25 |
申请人 |
CAMP ANNE MARIE;GALLAGHER PETER THADDEUS;LEDGARD ANDREW JAMES;SANDERSON ADAM JAN;COATES DAVID ANDREW;ELI LILLY AND COMPANY |
发明人 |
CAMP ANNE MARIE;GALLAGHER PETER THADDEUS;LEDGARD ANDREW JAMES;SANDERSON ADAM JAN;COATES DAVID ANDREW |
分类号 |
A61K31/5517;A61P25/20;C07D487/04 |
主分类号 |
A61K31/5517 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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