发明名称 HETEROARYLS AND USES THEREOF
摘要 This invention provides compounds of formula IA-a or IB-a and subsets thereof: wherein Z, HY, R1, R2, G1, W, n, and A and subsets thereof are as described in the specification. The compounds are inhibitors of PI3K and are thus useful for treating proliferative, inflammatory, or cardiovascular disorders.
申请公布号 US2012178723(A1) 申请公布日期 2012.07.12
申请号 US201113207696 申请日期 2011.08.11
申请人 HIROSE MASAAKI;HU ZHIGEN;HU YONGBO;LEE HONG MYUNG;SHI ZHAN;VYSKOCIL STEPAN;XU TIANLIN;MILLENNIUM PHARMACEUTICALS, INC. 发明人 HIROSE MASAAKI;HU ZHIGEN;HU YONGBO;LEE HONG MYUNG;SHI ZHAN;VYSKOCIL STEPAN;XU TIANLIN
分类号 A61K31/437;A61K31/381;A61K31/422;A61K31/4365;A61K31/4375;A61K31/4436;A61K31/4439;A61K31/4545;A61K31/4725;A61K31/496;A61K31/497;A61K31/498;A61K31/501;A61K31/506;A61K31/5377;A61K31/655;A61P7/02;A61P9/00;A61P9/12;A61P29/00;A61P35/00;A61P37/06;A61P37/08;C07D409/04;C07D409/14;C07D413/04;C07D413/14;C07D417/04;C07D417/14;C07D421/04;C07D471/04;C07D491/107;C07D495/04 主分类号 A61K31/437
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