发明名称 |
HETEROARYLS AND USES THEREOF |
摘要 |
This invention provides compounds of formula IA-a or IB-a and subsets thereof: wherein Z, HY, R1, R2, G1, W, n, and A and subsets thereof are as described in the specification. The compounds are inhibitors of PI3K and are thus useful for treating proliferative, inflammatory, or cardiovascular disorders.
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申请公布号 |
US2012178723(A1) |
申请公布日期 |
2012.07.12 |
申请号 |
US201113207696 |
申请日期 |
2011.08.11 |
申请人 |
HIROSE MASAAKI;HU ZHIGEN;HU YONGBO;LEE HONG MYUNG;SHI ZHAN;VYSKOCIL STEPAN;XU TIANLIN;MILLENNIUM PHARMACEUTICALS, INC. |
发明人 |
HIROSE MASAAKI;HU ZHIGEN;HU YONGBO;LEE HONG MYUNG;SHI ZHAN;VYSKOCIL STEPAN;XU TIANLIN |
分类号 |
A61K31/437;A61K31/381;A61K31/422;A61K31/4365;A61K31/4375;A61K31/4436;A61K31/4439;A61K31/4545;A61K31/4725;A61K31/496;A61K31/497;A61K31/498;A61K31/501;A61K31/506;A61K31/5377;A61K31/655;A61P7/02;A61P9/00;A61P9/12;A61P29/00;A61P35/00;A61P37/06;A61P37/08;C07D409/04;C07D409/14;C07D413/04;C07D413/14;C07D417/04;C07D417/14;C07D421/04;C07D471/04;C07D491/107;C07D495/04 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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