发明名称 |
PROCESS FOR PREPARING A 2-ALKYNYL SUBSTITUTED 5-AMINO-PYRAZOLO-[4,3-e]-1,2,4-TRIAZOLO[1,5-c]PYRIMIDINE |
摘要 |
A process for preparing 7-[2-[4-(6-fluoro-3-methyl-1,2-benzisoxazol-5-yl)-1-piperazinyl]ethyl]-2-(1-propynyl)-7H-pyrazolo-[4,3-e]-[1,2,4]-triazolo[1,5-c]pyrimidin-5-amine, intermediates useful in that process, and processes for preparing said intermediates are disclosed. |
申请公布号 |
EP2462144(A2) |
申请公布日期 |
2012.06.13 |
申请号 |
EP20100739457 |
申请日期 |
2010.08.03 |
申请人 |
SCHERING CORPORATION |
发明人 |
KUO, SHEN-CHUN;CHEN, YONGGANG;ECKERT, JEFFREY, M.;LEONG, WILLIAM, W.;ZOU, NANFEI;KUKLIS, GABRIEL, C. |
分类号 |
C07D487/14;A61K31/519;A61P25/28;C07C251/48;C07D231/38;C07D261/20;C07D403/04;C07D413/14 |
主分类号 |
C07D487/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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