发明名称 AMORPHOUS ATORVASTATIN CALCIUM OR PRAVASTATIN SODIUM HMG-COA REDUCTASE INHIBITORS OF DESIRED PARTICLE SIZE
摘要 A process for the preparation of amorphous HMG-CoA reductase inhibitor and its hydrates thereof of desired particle size, which comprises: (a) dissolving the HMG-CoA reductase inhibitor in a hydroxylic solvent; (b) removing the solvent by freeze-drying.
申请公布号 CA2479005(C) 申请公布日期 2012.05.22
申请号 CA20022479005 申请日期 2002.03.18
申请人 BIOCON LIMITED 发明人 POORNAPRAJNA, ACHARYA;MATHEW, JOY;CHANDRAPPA, RAVINDRA;SRIDHARAN, MADHAVAN;GANESH, SAMBASIVAM
分类号 C07D207/34;A61K31/22;A61K31/40;A61P3/06;C07C;C07C51/43;C07C59/62;C07C67/48;C07C67/52;C07C69/33;C07C69/732 主分类号 C07D207/34
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