发明名称 PROCESS FOR PREPARING AMINOCYCLOHEXYL ETHER COMPOUNDS
摘要 <p>The present invention relates to a process for preparing aminocyclohexyl ether compounds of Formula I: or the pharmaceutically acceptable salts and esters thereof. In particular, the instant invention is directed towards a process for preparing (1R,2R)-2-[(3R)-Hydroxypyrrolidinyl]-1-(3,4-dimethoxyphenethoxy)-cyclohexane as well as various intermediates.</p>
申请公布号 WO2012024100(A2) 申请公布日期 2012.02.23
申请号 WO2011US46885 申请日期 2011.08.08
申请人 MERCK SHARP & DOHME CORP.;LIMANTO, JOHN;BEUTNER, GREGORY, L.;YIN, JINGJUN;KLAPARS, ARTIS;ASHLEY, ERIC, R.;STROTMAN, HALLENA, R.;TRUPPO, MATTHEW, D.;CHUNG, CHEOL, K.;HUGHES, GREGORY;LIU, ZHIJIAN;GRAU, BRENDAN;JANEY, JACOB 发明人 LIMANTO, JOHN;BEUTNER, GREGORY, L.;YIN, JINGJUN;KLAPARS, ARTIS;ASHLEY, ERIC, R.;STROTMAN, HALLENA, R.;TRUPPO, MATTHEW, D.;CHUNG, CHEOL, K.;HUGHES, GREGORY;LIU, ZHIJIAN;GRAU, BRENDAN;JANEY, JACOB
分类号 C07D207/12 主分类号 C07D207/12
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