发明名称 PHTHALAZINONE KETONE DERIVATIVE, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL USE THEREOF
摘要 A phthalazinone ketone derivative as represented by formula (I), a preparation method thereof, a pharmaceutical composition containing the derivative, a use thereof as a poly (ADP-ribose) polymerase (PARP) inhibitor, and a cancer treatment method thereof.
申请公布号 WO2012019427(A1) 申请公布日期 2012.02.16
申请号 WO2011CN01223 申请日期 2011.07.26
申请人 SHANGHAI HENGRUI PHARMACEUTICAL CO., LTD.;JIANGSU HENGRUI MEDICINE CO., LTD.;TANG, PENGCHO;LI, XIN;LI, XIANGQIN;CHEN, YANG;WANG, BIN;ZHU, ZHE 发明人 TANG, PENGCHO;LI, XIN;LI, XIANGQIN;CHEN, YANG;WANG, BIN;ZHU, ZHE
分类号 C07D487/04;A61K31/502;A61K31/5025;A61P35/00;A61P43/00;C07D403/12 主分类号 C07D487/04
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