发明名称 |
SYNTHESIS OF BORONIC ESTER AND ACID COMPOUNDS |
摘要 |
THE INVENTION RELATES TO THE SYNTHESIS OF BOIONIC ESTER AND ACID COMPOUNDS. MORE PARTICULARLY, THE INVENTION PROVIDES IMPROVED SYNTHETIC PROCESSES FOR THE LARGE-SCALE PRODUCTION OF BORONIC ESTER AND ACID COMPOUNDS, INCLUDING THE PEPTIDE BORONIC ACID PROTEASOME INHIBITOR BORTEZOMIB. |
申请公布号 |
MY145427(A) |
申请公布日期 |
2012.02.15 |
申请号 |
MY2005PI01304 |
申请日期 |
2005.03.24 |
申请人 |
MILLENNIUM PHARMACEUTICALS, INC. |
发明人 |
FRASER PICKERSGILL;FANG-TING CHIU;VITHALANAND R. KULKARNI;JOHN BISHOP;CHRISTOPH KOELLNER;JEAN-MARCH GOMEZ;ACHIM GEISER;ROBERT HETT;VINCE AMMOSCATO;STEVEN MUNK;YOUNG LO |
分类号 |
C07F5/02;C07F5/04 |
主分类号 |
C07F5/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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