发明名称 DIHYDROPYRAZOLOPYRIMIDINONE DERIVATIVES
摘要 <p>63 - DIHYDROPYRAZOLOPYRIMIDINONE DERIVATIVES ABSTRACT THE INVENTION RELATES TO COMPOUNDS OF A GENERAL FORMULA (1): R1 2 R RS R6 0 AL H WHEREIN AI IS SELECTED FROM THE FOLLOWING FORMULA (AAL): -N /--J NR'C -CNR'C (AAL RI IS A LOWER ALKENYL GROUP OR A LOWER ALKYNYL GROUP; R2 IS A PHENYL, PYRIDYL OR THIENYL GROUP; R5 AND R6 ARE A HVDROGEN ATOM, A LOWER ALKYL 10 GROUP OR A HYDROXY-LOWER ALKYL GROUP, ETC. 'ME COMPOUNDS OF THE INVENTION HAVE EXCELLENT WEEL KINASE-INHIBITORY EFFECT AND ARE THEREFORE USEFUL IN THE FIELD OF MEDICINES, ESPECIALLY TREATMENT OF VARIOUS CANCERS. (NO</p>
申请公布号 MY145408(A) 申请公布日期 2012.02.15
申请号 MY2008PI03651 申请日期 2008.09.18
申请人 MSD K.K. 发明人 SAKAMOTO, TOSHIHIRO;NISHIBATA, TOSHIHIDE;YOSHIZUMI, TAKASHI;HIRAI, HIROSHI;SUNAMI, SATOSHI;YAMAMOTO, FUYUKI;NIIYAMA, KENJI;BAMBA, MAKOTO;TAKAHASHI, KEIJI;FURUYAMA, HIDETOMO;SAGARA, TAKESHI;OTSUKI, SACHIE
分类号 C07D487/04 主分类号 C07D487/04
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