发明名称 Molecular Crystal of (4-(1,8-Naphthyridin-2-YL)Piperidin-1-YL)Pyrimidine Derivative
摘要 A molecular crystal form of (S)-3-(2,5-dimethyl-6-(4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)piperidin-1-yl)pyrimidin-4-ylamino)-2-(4-methoxyphenylsulfonamido)propanoic acid is characterized by an X-ray powder diffraction (“XRPD”) spectrum that comprises peaks at 2&thetas; angles of 7.44, 14.80, 16.64, and 23.04±0.2°. The molecular crystal can be formulated into pharmaceutical composition for treating or controlling diseases resulting from pathological angiogenesis.
申请公布号 US2011237605(A1) 申请公布日期 2011.09.29
申请号 US201113018896 申请日期 2011.02.01
申请人 PHILLIPS ERIC;SHAWER MOHANNAD 发明人 PHILLIPS ERIC;SHAWER MOHANNAD
分类号 A61K31/506;A61P27/02;A61P35/00;C07D471/04 主分类号 A61K31/506
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