发明名称 |
1,3,4,8-TETRAHYDRO-2H-PYRIDO[1,2-A]PYRAZINE DERIVATIVE AND USE OF SAME AS HIV INTEGRASE INHIBITOR |
摘要 |
<p>Disclosed is a novel 1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine derivative, a pharmaceutically acceptable salt thereof or a solvate thereof, which is useful as an anti-HIV agent. Specifically disclosed is a compound represented by general formula (I), a pharmaceutically acceptable salt thereof or a solvate thereof. (In the formula, the symbols are as defined in the description.)</p> |
申请公布号 |
WO2011105590(A1) |
申请公布日期 |
2011.09.01 |
申请号 |
WO2011JP54404 |
申请日期 |
2011.02.25 |
申请人 |
JAPAN TOBACCO INC.;MIYAZAKI, SUSUMU;BESSHO, YUKI;ADACHI, KAORU;KAWASHITA, SEIJI;ISOSHIMA, HIROTAKA;OSHITA, KENGO;FUKUDA, SHUNICHI |
发明人 |
MIYAZAKI, SUSUMU;BESSHO, YUKI;ADACHI, KAORU;KAWASHITA, SEIJI;ISOSHIMA, HIROTAKA;OSHITA, KENGO;FUKUDA, SHUNICHI |
分类号 |
C07D471/04;A61K31/4985;A61K31/5377;A61P31/18;A61P43/00 |
主分类号 |
C07D471/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|