发明名称 PROCESS FOR PREPARATION OF PROPARGYLATED AMINOINDANS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF
摘要 A process for preparation of propargylated aminoindans or pharmaceutically acceptable salts thereof, comprises: a) reacting an indanone derivative or a salt thereof with propargyl amine or a salt thereof in the presence of a Lewis acid; b) subjecting the resultant reaction mixture to reduction.
申请公布号 WO2011048612(A3) 申请公布日期 2011.08.11
申请号 WO2010IN00671 申请日期 2010.10.08
申请人 GLENMARK GENERICS LIMITED;THANEDAR, AMIT, ANANT;DESHMUKH, SHEKHAR, ASHOK;ZOPE, SUNIL, SUDHAKAR;KELKAR, LAXMIKANT, MADHUKAR;KOILPILLAI, JOSEPH, PRABAHAR;GAJERA, JITENDRA, MAGANBHAI 发明人 THANEDAR, AMIT, ANANT;DESHMUKH, SHEKHAR, ASHOK;ZOPE, SUNIL, SUDHAKAR;KELKAR, LAXMIKANT, MADHUKAR;KOILPILLAI, JOSEPH, PRABAHAR;GAJERA, JITENDRA, MAGANBHAI
分类号 C07C211/42;A61K31/135;A61P25/16;C07C209/22;C07C269/06;C07C271/44 主分类号 C07C211/42
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