发明名称 |
MALEATE CO-CRYSTAL OF AZD1152 AND USE THEREOF FOR THE TREATMENT OF CANCER |
摘要 |
The present invention relates to a novel co-crystal of 2-(ethyl[3-( {4-[(5- {2-[(3-fluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]quinazolin-7-yl}oxy)propyl]amino} ethyl dihydrogen phosphate (AZD1152) which is an aurora kinase inhibitor that is useful in the treatment of hyperproliferative diseases such as cancer. |
申请公布号 |
UA95108(C2) |
申请公布日期 |
2011.07.11 |
申请号 |
UA20080013934 |
申请日期 |
2007.05.14 |
申请人 |
ASTRAZENECA AB |
发明人 |
SEPENDA GEORGE JOSEPH;STOREY RICHARD |
分类号 |
C07D403/12;A61K31/661;C07F9/09 |
主分类号 |
C07D403/12 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|