发明名称 |
PIPERIDINE DERIVATIVE AND ITS USE FOR THE TREATMENT OF DIABETS AND OBESITY |
摘要 |
<p>The present invention relates to the GPR119 agonist, N-(2-fluoro-4-(methylsulfonyl)phenyl)-5-methyl-6-(1-(5-methylpyrazin-2-yl)piperidin-4-yloxy)pyrimidin-4-amine (Compound 1, Formula (I)), and pharmaceutically acceptable salts, solvates, and hydrates thereof, that are useful in the treatment of GPR119-related disorders, such as, metabolic-related disorders and complications thereof, such as, diabetes and obesity.</p> |
申请公布号 |
WO2011005929(A1) |
申请公布日期 |
2011.01.13 |
申请号 |
WO2010US41325 |
申请日期 |
2010.07.08 |
申请人 |
ARENA PHARMACEUTICALS, INC.;JONES, ROBERT M.;LEHMANN, JUERG |
发明人 |
JONES, ROBERT M.;LEHMANN, JUERG |
分类号 |
C07D403/14;A61K31/506;A61P3/04;A61P3/10 |
主分类号 |
C07D403/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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