发明名称 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS
摘要 The present invention relates to sulfamoyl benzoic acid derivatives of formula (I) or a pharmaceutically acceptable salt thereof, processes for their preparation, pharmaceutical compositions containing them and their use in the treatment of various disorders which are mediated via the TRPM8 receptor.
申请公布号 CA2757761(A1) 申请公布日期 2010.11.04
申请号 CA20102757761 申请日期 2010.05.06
申请人 RAQUALIA PHARMA INC. 发明人 INOUE, TADASHI;OHMI, MASASHI;KAWAMURA, KIYOSHI;ANDO, KAZUO;SHISHIDO, YUJI
分类号 A61K31/18;A61K31/196;A61K31/44;A61K31/443;A61K31/4436;A61K31/4439;A61K31/444;A61K31/4453;A61K31/4709;A61K31/495;A61K31/5375;A61K31/5377;A61P1/04;A61P9/10;A61P11/06;A61P13/00;A61P13/02;A61P13/08;A61P13/10;A61P13/12;A61P19/08;A61P25/00;A61P25/04;A61P25/22;A61P25/24;A61P29/00;A61P43/00;C07C311/21;C07C311/29;C07D211/16;C07D213/42;C07D213/76;C07D295/12;C07D295/18;C07D401/12;C07D401/14;C07D405/04;C07D405/12;C07D409/04;C07D409/12;C07D413/12;C07D417/12 主分类号 A61K31/18
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