发明名称 |
SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS |
摘要 |
The present invention relates to sulfamoyl benzoic acid derivatives of formula (I) or a pharmaceutically acceptable salt thereof, processes for their preparation, pharmaceutical compositions containing them and their use in the treatment of various disorders which are mediated via the TRPM8 receptor.
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申请公布号 |
CA2757761(A1) |
申请公布日期 |
2010.11.04 |
申请号 |
CA20102757761 |
申请日期 |
2010.05.06 |
申请人 |
RAQUALIA PHARMA INC. |
发明人 |
INOUE, TADASHI;OHMI, MASASHI;KAWAMURA, KIYOSHI;ANDO, KAZUO;SHISHIDO, YUJI |
分类号 |
A61K31/18;A61K31/196;A61K31/44;A61K31/443;A61K31/4436;A61K31/4439;A61K31/444;A61K31/4453;A61K31/4709;A61K31/495;A61K31/5375;A61K31/5377;A61P1/04;A61P9/10;A61P11/06;A61P13/00;A61P13/02;A61P13/08;A61P13/10;A61P13/12;A61P19/08;A61P25/00;A61P25/04;A61P25/22;A61P25/24;A61P29/00;A61P43/00;C07C311/21;C07C311/29;C07D211/16;C07D213/42;C07D213/76;C07D295/12;C07D295/18;C07D401/12;C07D401/14;C07D405/04;C07D405/12;C07D409/04;C07D409/12;C07D413/12;C07D417/12 |
主分类号 |
A61K31/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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