发明名称 |
PYRROLOPYRAZOLE, POTENT KINASE INHIBITORS |
摘要 |
Pyrrole pyrazole compounds of formula I, compositions including these compounds and methods of their use are provided. Preferred compounds of formula I have activity as protein kinase inhibitors, including as inhibitors of PAK4.
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申请公布号 |
US2010222342(A1) |
申请公布日期 |
2010.09.02 |
申请号 |
US20050813658 |
申请日期 |
2005.12.28 |
申请人 |
ZHANG JUNHU;GUO CHUANGXING;BOUZIDA DJAMAL;DONG LIMING;LI HAITAO;MARAKOVITS JOSEPH TIMOTHY;YANG ANLE;HONG YUFENG |
发明人 |
ZHANG JUNHU;GUO CHUANGXING;BOUZIDA DJAMAL;DONG LIMING;LI HAITAO;MARAKOVITS JOSEPH TIMOTHY;YANG ANLE;HONG YUFENG |
分类号 |
A61K31/5377;A61K31/4439;A61K31/506;A61K31/517;A61K31/519;A61K31/53;A61P35/00;C07D239/47;C07D401/14;C07D403/14;C07D413/14;C07D491/048;C07D495/04 |
主分类号 |
A61K31/5377 |
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