发明名称 Radiolabeled cannabinoid-1 receptor modulators
摘要 The present invention relates to particular radiolabeled Cannabinoid-1 (CB1) receptor modulators, and methods of using these modulators for labeling and diagnostic imaging of Cannabinoid-1 receptors in mammals, particularly humans. In addition, intermediates useful for the synthesis of the radiolabeled Cannabinoid-1 receptor modulators are also disclosed, as well as the processes for synthesizing the radiolabeled Cannabinoid-1 receptor modulators. Still further, formulations of the radiolabeled Cannabinoid-1 receptor compounds are described.
申请公布号 US7754188(B2) 申请公布日期 2010.07.13
申请号 US20050559228 申请日期 2005.12.06
申请人 MERCK SHARP & DOHME CORP. 发明人 BURNS H. DONALD;CHEN ALEX M.;GIBSON RAYMOND E.;GOULET MARK T.;HAGMANN WILLIAM K.;HAMILL TERENCE G.;JEWELL JAMES P.;LIN LINUS S.;LIU PING;PERESYPKIN ANDREY V.
分类号 A61K51/00;A61K51/04;A61M36/14;C07D213/64;C07D239/34 主分类号 A61K51/00
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