发明名称 PROCESS FOR PRODUCTION OF QUINAZOLINE DERIVATIVE
摘要 Provided is a production method wherein two reaction steps for producing a target compound (III) from a methoxycarbonyl compound via a methoxyamide compound are continuously carried out to thereby conduct these reactions substantially in a single step. According to this method, the compound (III), which is useful as an intermediate in producing a dual tyrosine kinase inhibitor, can be conveniently produced at a high yield.
申请公布号 CA2745150(A1) 申请公布日期 2010.07.01
申请号 CA20092745150 申请日期 2009.12.24
申请人 SHIONOGI & CO., LTD. 发明人 HAGIHARA, MOTOYUKI;SHINOMOTO, SHOJI
分类号 C07D239/94 主分类号 C07D239/94
代理机构 代理人
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