发明名称 Process for the Preparation of Esomeprazole Magnesium Dihydrate
摘要 A process for preparing Form A of (S)-5-methoxy-2-[[(4-methoxy-3,5-dimethyl-2-pyridinyl)-methyl]sulfinyl]-1H-benzimidazole magnesium dihydrate, processes for preparing various intermediates useful in the preparation of Form A of (S)-5-methoxy-2-[[(4-methoxy-3,5-dimethyl-2-pyridinyl)-methyl]sulfinyl]-1H-benzimidazole magnesium dihydrate and a novel polymorphic Form II of 5-methoxy-2-[[(4-methoxy-3,5-dimethyl-2-pyridinyl)-methyl]thio]-1H-benzimidazole.
申请公布号 US2010113526(A1) 申请公布日期 2010.05.06
申请号 US20080527967 申请日期 2008.02.21
申请人 CIPLA LIMITED 发明人 RAO DHARMARAJ RAMACHANDRA;KANKAN RAJENDRA NARAYANRAO;PATHI SRINIVAS LAXMINARAYAN;BANGALORE GOPALAKRISHNA SUMANA
分类号 A61K31/4439;A61P1/04;C07D401/12 主分类号 A61K31/4439
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