发明名称 LOW MOLECULAR WEIGHT THYROID STIMULATING HORMONE RECEPTOR (TSHR) AGONISTS
摘要 Disclosed are oxo-hydroquinazolines of formula I that are useful as selective TSHR agonists. The compounds may be used for detecting or treating thyroid cancer, or treating a bone degenerative disorder.
申请公布号 CA2741030(A1) 申请公布日期 2010.04.29
申请号 CA20082741030 申请日期 2008.10.20
申请人 THE GOVERNMENT OF THE UNITED STATES OF AMERICA ASREPRESENTED BY THE SEC RETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES 发明人 GERSHENGORN, MARVIN, C.;NEUMANN, SUSANNE;RAAKA, BRUCE, M.;THOMAS, CRAIG, J.;INGLESE, JAMES;SOUTHALL, NOEL, T.;TITUS, STEVEN;ZHENG, WEI;HUANG, WENWEI;KRAUSE, GERD;KLEINAU, GUNNAR
分类号 C07D235/18;A61K31/4184 主分类号 C07D235/18
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