发明名称 |
SUBSTITUTED PYRAZOLE DERIVATIVE. |
摘要 |
<p>Disclosed are a novel pyrazole derivative and an androgen receptor antagonist containing the pyrazole derivative. Specifically disclosed is a compound represented by the formula (I') below or a salt thereof. (In the formula, R1 represents a hydrogen atom, a group having a carbon atom serving as a bonding hand, a group having a nitrogen atom serving as a bonding hand, a group having an oxygen atom serving as a bonding hand or a group having a sulfur atom serving as a bonding hand; R2 represents a phenyl group having a cyano (which may further have a substituent other than cyano); R3 represents a hydrogen atom, a group having a carbon atom serving as a bonding hand, a group having a nitrogen atom serving as a bonding hand, a group having an oxygen atom serving as a bonding hand or a group having a sulfur atom serving as a bonding hand; R4 represents an optionally substituted cyclic group; and X represents an optionally substituted methylene or CO.).</p> |
申请公布号 |
MX2010002266(A) |
申请公布日期 |
2010.03.25 |
申请号 |
MX20100002266 |
申请日期 |
2008.08.27 |
申请人 |
TAKEDA PHARMACEUTICAL COMPANY LIMITED |
发明人 |
MITSUHIRO ITO;TOMOHIKO SUZAKI;SATOSHI YAMAMOTO |
分类号 |
C07D231/12;A61K31/415;A61K31/4162;A61K31/4178;A61K31/4192;A61K31/4196;A61K31/42;A61K31/422;A61K31/427;A61K31/433;A61K31/4439;A61K31/4545;A61K31/4709;A61K31/497;A61K31/498;A61K31/506;A61K31/5377;A61P5/28;A61P13/08;A61P35/00;A61P43/00;C07D401/06;C07D401/10;C07D401/12;C07D403/06;C07D403/12;C07D405/06;C07D409/06;C07D409/14;C07D413/06;C07D417/06;C07D417/14;C07D495/04 |
主分类号 |
C07D231/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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