发明名称 NOVEL HYDROXAMIC ACID DERIVATIVE HAVING NAPHTHYRIDINE-N-OXIDE
摘要 <p>Provided is a novel compound useful as a pharmaceutical that exhibits strong antibacterial activity for gram negative bacteria, such as Pseudomonas aeruginosa, and for drug-resistant bacterial strains thereof, based on LpxC inhibitory activity. Provided is a hydroxamic acid derivative represented by general formula (1) or a pharmacologically permitted salt thereof. (1)</p>
申请公布号 WO2010024356(A1) 申请公布日期 2010.03.04
申请号 WO2009JP65006 申请日期 2009.08.27
申请人 TAISHO PHARMACEUTICAL CO., LTD.;TOYAMA CHEMICAL CO., LTD.;TAKASHIMA, HAJIME;SUGA, YOICHIRO;URABE, HIROKI;TSURUTA, RISA;KOTSUBO, HIRONORI;OOHORI, RYUTARO;KAWAGUCHI, YASUKO 发明人 TAKASHIMA, HAJIME;SUGA, YOICHIRO;URABE, HIROKI;TSURUTA, RISA;KOTSUBO, HIRONORI;OOHORI, RYUTARO;KAWAGUCHI, YASUKO
分类号 A61K31/4375;C07D471/04;A61P31/04;A61P43/00 主分类号 A61K31/4375
代理机构 代理人
主权项
地址