发明名称 HIV INTEGRASE INHIBITORS
摘要 <p>Tricyclic compounds of Formula I are inhibitors of HIV integrase and inhibitors of HIV replication: (I) wherein G, T, R1, R2, R3A, R3B, R4A, R4B, R5A, R5B, R6A and R6B are defined herein. The compounds are useful for the prophylaxis or treatment of infection by HIV and the prophylaxis, treatment, or delay in the onset or progression of AIDS. The compounds are employed against HIV infection and AIDS as compounds per se (or as hydrates or solvates thereof) or in the form of pharmaceutically acceptable salts. The compounds and their salts can be employed as ingredients in pharmaceutical compositions, optionally in combination with other antivirals, immunomodulators, antibiotics or vaccines.</p>
申请公布号 WO2009154870(A1) 申请公布日期 2009.12.23
申请号 WO2009US41598 申请日期 2009.04.24
申请人 MERCK & CO., INC.;ISAACS, RICHARD, C. A.;WAI, JOHN, S.;FISHER, THORSTEN, E. 发明人 ISAACS, RICHARD, C. A.;WAI, JOHN, S.;FISHER, THORSTEN, E.
分类号 A01N43/00;A61K31/553;A61K31/554 主分类号 A01N43/00
代理机构 代理人
主权项
地址