发明名称 PROCESS FOR PREPARING POSACONAZOLE AND INTERMEDIATES THEREOF
摘要 The present invention relates to an industrially advantageous process for the preparation of tetrahydrofuran antifungals preferably posaconazole of formula I. The present invention further relates to improved processes for preparing key and novel intermediates useful in the preparation of posaconazole. The present invention further relates to improved processes for preparing the compound of formula II, a key intermediate in the preparation of posaconazole.
申请公布号 WO2009141837(A2) 申请公布日期 2009.11.26
申请号 WO2009IN00292 申请日期 2009.05.19
申请人 IND-SWIFT LABORATORIES LIMITED;CHIDAMBARAM, VENKATESWARAN, SRINIVASAN;MIRYALA, ATCHUTA, KISHORE;WADHWA, LALIT 发明人 CHIDAMBARAM, VENKATESWARAN, SRINIVASAN;MIRYALA, ATCHUTA, KISHORE;WADHWA, LALIT
分类号 C07D405/14 主分类号 C07D405/14
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