发明名称 |
COMPOUND HAVING NPY Y5 RECEPTOR ANTAGONIST ACTIVITY |
摘要 |
<p>Disclosed is a novel compound having NPY Y5 receptor antagonist activity, specifically a compound represented by formula (I), a pharmaceutically acceptable salt thereof, or a solvate of the compound or the salt. [In the formula, R1 represents a substituted or unsubstituted alkyl or the like; R2 represents a hydrogen, or a substituted or unsubstituted alkyl; ring A represents a monocyclic or bicyclic aromatic heterocycle; R3 represents a substituted or unsubstituted aryl, a substituted or unsubstituted heteroaryl, or a substituted or unsubstituted heterocyclyl; R4 represents a halogen, a cyano, a substituted or unsubstituted alkyl, a substituted or unsubstituted cycloalkyl or the like; m represents an integer of 0-2; n represents an integer of 0-5; R represents a halogen, an oxo, a cyano, a substituted or unsubstituted alkyl or the like; and p represents an integer of 0-2.]</p> |
申请公布号 |
WO2009131096(A1) |
申请公布日期 |
2009.10.29 |
申请号 |
WO2009JP57856 |
申请日期 |
2009.04.20 |
申请人 |
SHIONOGI & CO., LTD.;SAKAGAMI, MASAHIRO;HASHIZUME, HIROSHI;TANAKA, SATORU;OKUNO, TAKAYUKI;YARI, HIROSHI;TONOGAKI, KEISUKE;KOUYAMA, NAOKI |
发明人 |
SAKAGAMI, MASAHIRO;HASHIZUME, HIROSHI;TANAKA, SATORU;OKUNO, TAKAYUKI;YARI, HIROSHI;TONOGAKI, KEISUKE;KOUYAMA, NAOKI |
分类号 |
C07D207/335;A61K31/40;A61K31/4045;A61K31/415;A61K31/416;A61K31/4164;A61K31/4178;A61K31/4196;A61K31/422;A61K31/427;A61K31/437;A61K31/4439;A61K31/444;A61K31/451;A61K31/4545;A61K31/497;A61K31/4985;A61K31/506;A61K31/519;A61K31/5377;A61P1/14;A61P3/04;A61P9/00;A61P9/04;A61P9/12;A61P15/08;A61P15/10;A61P25/08;A61P25/20;A61P43/00;C07D209/14;C07D211/40;C07D231/12;C07D231/14;C07D233/64;C07D249/08;C07D401/04;C07D401/14;C07D403/04;C07D407/04;C07D413/04;C07D417/04;C07D471/04;C07D487/04 |
主分类号 |
C07D207/335 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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