发明名称 Polypeptides having anti-HIV activity and compositions comprising same
摘要 The present invention relates to a polypeptide represented by the formula: <?in-line-formulae description="In-line Formulae" end="lead"?>A1-Arg-A2-Cys-Tyr-A3-A4-X-A5-A6-Cit-Cys-A7 (I)<?in-line-formulae description="In-line Formulae" end="tail"?> (wherein A1 represents a hydrogen atom or an arginine, lysine, ornithine, citrulline, alanine residue, etc.; A2 represents an aromatic amino acid residue; A3, A4 and A6 represent an arginine, lysine, ornithine, citrulline or alanine residue, A5 represents a tyrosine, phenylalanine, alanine, naphthylalanine or citrulline residue; A7 represents a lysine or arginine residue in which a carboxyl group may be amidated; X represents a D-ornithyl-proline, prolyl-D-ornithine, D-lysyl-proline residue, etc.; provided that either of A1, A3, A4, A5, A6 and A7 is an alanine residue, etc., or X is citrulline, etc.) or a salt thereof.
申请公布号 US7595298(B2) 申请公布日期 2009.09.29
申请号 US20060497225 申请日期 2006.08.01
申请人 BIOKINE THERAPEUTICS LTD. 发明人 FUJII NOBUTAKA
分类号 A61K38/00;A61K39/12;A61K39/21;A61P31/18;C07K2/00;C07K4/00;C07K5/00;C07K7/08;C07K14/00;C07K14/435;C07K16/00;C07K17/00 主分类号 A61K38/00
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