发明名称 Crystalline forms of mc4r agonist and process for synthesis
摘要 The present invention relates to a process for producing N-{(1S)-1-[2-(1-{[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl]carbonyl}piperidin-4-yl)-5-chlorophenyl]ethyl}acetamide, and novel crystalline salts, hydrates, solvates, and polymorphic forms thereof.
申请公布号 US2009233967(A1) 申请公布日期 2009.09.17
申请号 US20060921824 申请日期 2006.06.23
申请人 CALABRIA RALPH;CHENG YU;FERLITA RUSSELL R;KAMALI ASHKAN;MURRY JERRY A;MATHRE DAVID;PERESYPKIN ANDREY V;THOMPSON KAREN;WANG JIAN;WENSLOW ROBERT M 发明人 CALABRIA RALPH;CHENG YU;FERLITA RUSSELL R.;KAMALI ASHKAN;MURRY JERRY A.;MATHRE DAVID;PERESYPKIN ANDREY V.;THOMPSON KAREN;WANG JIAN;WENSLOW ROBERT M.
分类号 A61K31/454;C07D401/06 主分类号 A61K31/454
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