发明名称 BENZAMIDE DERIVATIVE
摘要 PROBLEM TO BE SOLVED: To provide a novel benzamide derivative having a vasopressin antagonistic activity or the like. SOLUTION: The novel benzamide derivative is represented by formula (I) (wherein R<SP>1</SP>is an aryl optionally substituted with a lower alkoxy or the like; R<SP>2</SP>is a lower alkyl or the like, R<SP>3</SP>is hydrogen or the like; A is NH or the like; E is -C(=O)- or the like; X is -CH=CH-, -CH=N- or S; and Y is a condensed heterocyclic group or the like). COPYRIGHT: (C)2009,JPO&INPIT
申请公布号 JP2009143904(A) 申请公布日期 2009.07.02
申请号 JP20080305474 申请日期 2008.10.31
申请人 ASTELLAS PHARMA INC 发明人 SETOI HIROYUKI;OKAWA TAKEHIKO;YOSHIMITSU TATSUYA;SAWADA HITOSHI;SAWADA YUKI;OKU TERUO
分类号 C07C237/44;A61K31/166;A61K31/40;A61K31/4035;A61K31/41;A61K31/415;A61K31/4184;A61K31/421;A61K31/422;A61K31/423;A61K31/454;A61K31/495;A61K31/496;A61K31/497;A61K31/498;A61K31/517;A61K31/52;A61K31/535;A61K31/5375;A61K31/5377;A61P1/08;A61P1/16;A61P3/10;A61P7/00;A61P7/10;A61P9/00;A61P9/10;A61P9/12;A61P13/12;A61P25/20;A61P43/00;C07C231/12;C07C237/42;C07D209/02;C07D209/08;C07D209/12;C07D209/14;C07D209/26;C07D209/34;C07D209/40;C07D209/42;C07D209/48;C07D215/48;C07D231/56;C07D235/06;C07D235/08;C07D235/10;C07D235/12;C07D235/14;C07D235/16;C07D235/24;C07D235/26;C07D235/28;C07D235/30;C07D235/32;C07D239/88;C07D239/96;C07D241/42;C07D249/18;C07D263/10;C07D263/30;C07D263/54;C07D263/56;C07D265/32;C07D265/34;C07D295/12;C07D295/135;C07D295/18;C07D295/185;C07D401/04;C07D401/06;C07D401/12;C07D403/04;C07D403/06;C07D403/12;C07D413/12;C07D471/04;C07D473/00;C07D487/04;C07D521/00;C07F7/18 主分类号 C07C237/44
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