发明名称 CHIRAL SYNTHESIS OF DIAZEPINOQUINOLINES
摘要 The present invention relates to improved methods of resolution and recrystallization for synthesizing compounds of formulae (I-1) or (A) useful as 5HT2 agonists or partial agonists, including intermediates thereto.
申请公布号 WO2009039362(A3) 申请公布日期 2009.04.30
申请号 WO2008US77003 申请日期 2008.09.19
申请人 WYETH;MEGATI, SREENIVASULU;BHANSALI, SHILPA;DEHNHARDT, CHRISTOPH;DESHMUKH, SUBODH;FUNG, PETER;MACEWAN, MICHAEL;TINDER, ROBERT, J. 发明人 MEGATI, SREENIVASULU;BHANSALI, SHILPA;DEHNHARDT, CHRISTOPH;DESHMUKH, SUBODH;FUNG, PETER;MACEWAN, MICHAEL;TINDER, ROBERT, J.
分类号 C07D471/06;A61K31/5517;A61P25/18 主分类号 C07D471/06
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